SCHEMBL6559990

SCHEMBL6559990

Nc1ccc2nc(N3CC4CCCCCCCCCCCCCCCCCCCCCC3CC4)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.43
HRH3 Q9Y5N1 9/20 0.41
KDM4E B2RXH2 5/20 0.39
MAPT P10636 2/20 0.39
GFER P55789 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
PLAU P00749 1/20 0.39
BACE1 P56817 1/20 0.37
LMNA P02545 2/20 0.37
POLB P06746 1/20 0.37
CASP6 P55212 1/20 0.37
MEN1 O00255 1/20 0.36
RGS12 O14924 1/20 0.36
NPC1 O15118 1/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
KEAP1 Q14145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5873493 0.94 MCHR1 (0.46) MCHR1HRH3KDM4EMAPTALDH1A1
SCHEMBL6558013 0.80 ALDH1A1 (0.49) MCHR1MAPTALDH1A1LMNAPOLB
SCHEMBL4847239 0.74 CHRNA7 (0.46) KDM4ELMNAPOLBCASP6
SCHEMBL5873479 0.72 ALDH1A1 (0.54) MCHR1ALDH1A1LMNA
SCHEMBL5873568 0.69 MAP4K4 (0.51) HRH3KDM4EALDH1A1PLAULMNA
SCHEMBL6559810 0.69 MCHR1 (0.42) MCHR1HRH3PLAU
SCHEMBL5873732 0.68 MCHR1 (0.43) MCHR1HRH3
SCHEMBL6557970 0.66 MCHR1 (0.59) MCHR1HRH3
SCHEMBL29209061 0.65 KDM4E (0.50) HRH3KDM4EALDH1A1TDP1PLAU
SCHEMBL5873634 0.65 MCHR1 (0.75) MCHR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450801-A2 2-AMINOQUINOLINE COMPOUNDS Merck & Co., Inc. (US) 2004-09-01 EP disclosed
WO-2003045313-A2 2-AMINOQUINOLINE COMPOUNDS MERCK & CO. INC. (US) 2003-06-05 WO disclosed