SCHEMBL6558533

SCHEMBL6558533

[O]C(=O)n1cc2ccccc2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.35
ALOX12 P18054 1/20 0.35
CES2 O00748 2/20 0.34
CES1 P23141 2/20 0.34
NOTUM Q6P988 1/20 0.34
ALDH1A1 P00352 4/20 0.33
KMT2A Q03164 2/20 0.33
DAO P14920 2/20 0.33
NR4A2 P43354 2/20 0.33
NR4A1 P22736 1/20 0.33
NR4A3 Q92570 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TSHR P16473 3/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075524 0.79 ALDH1A1 (0.38) CYP2A6ALOX12CES2CES1ALDH1A1
SCHEMBL15880060 0.77 NOTUM (0.47) CES2CES1NOTUMALDH1A1KMT2A
SCHEMBL3700594 0.77 TSHR (0.39) CYP2A6ALOX12NOTUMALDH1A1KMT2A
SCHEMBL9956507 0.77 CES2 (0.38) CYP2A6ALOX12CES2CES1NOTUM
Hydrochloric Acid SCHEMBL28200481 0.75 TSHR (0.38) ALDH1A1KMT2AKDM4EMEN1HPGD
SCHEMBL8768144 0.73 HPGD (0.34) CES2CES1NOTUMALDH1A1KMT2A
SCHEMBL3172447 0.73 TSHR (0.50) CES2CES1ALDH1A1KMT2ADAO
SCHEMBL23723572 0.72 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1RAB9A
SCHEMBL28323036 0.72 P2RX4 (0.44) ALDH1A1KMT2ANR4A2KDM4EMEN1
SCHEMBL17797526 0.72 CES1 (0.40) CES1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998488-B1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-03-17 EP disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed
EP-0998488-A1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2000-05-10 EP disclosed
WO-1999002549-A1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-01-21 WO disclosed