SCHEMBL6558665

SCHEMBL6558665

CN(C)c1ccc(C(c2ccc(N(C)C)cc2)c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
LMNA P02545 3/20 0.50
TP53 P04637 2/20 0.50
ATM Q13315 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HTT P42858 2/20 0.46
MEN1 O00255 2/20 0.45
SLC2A1 P11166 1/20 0.43
ALDH1A1 P00352 5/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK1 P28482 1/20 0.40
PHLPP2 Q6ZVD8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558728 0.86 ALDH1A1 (0.43) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL9657128 0.83 KMT2A (0.44) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL3902654 0.82 KMT2A (0.54) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL8777757 0.82 CYP3A4 (0.48) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL6558704 0.81 SLC2A1 (0.42) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL5011743 0.79 SLC2A1 (0.59) KMT2ATP53MEN1SLC2A1ALDH1A1
SCHEMBL6557047 0.79 SLC2A1 (0.46) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL6557998 0.79 SLC2A1 (0.46) KMT2ALMNAATMSMN1; SMN2NPSR1
SCHEMBL30327120 0.79 LMNA (0.40) KMT2ALMNATP53ATMSMN1; SMN2
SCHEMBL5555851 0.77 KMT2A (0.47) KMT2ALMNATP53ATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100483-B1 GLUCOCORTICOID-SELECTIVE ANTI-INFLAMMATORY AGENTS ABBOTT LAB (US) 2004-09-29 EP claimed
EP-3324242-B1 INTERMEDIATE TRANSFER MEMBER, METHOD FOR PRODUCING INTERMEDIATE TRANSFER MEMBER, AND IMAGE FORMING APPARATUS KONICA MINOLTA INC (JP) 2020-06-17 EP disclosed
US-10274874-B2 Intermediate transfer member, method for producing intermediate transfer member, and image forming apparatus Konica Minolta, Inc. (JP) 2019-04-30 US disclosed
EP-3324242-A1 INTERMEDIATE TRANSFER MEMBER, METHOD FOR PRODUCING INTERMEDIATE TRANSFER MEMBER, AND IMAGE FORMING APPARATUS Konica Minolta, Inc. (JP) 2018-05-23 EP disclosed
US-20180136590-A1 INTERMEDIATE TRANSFER MEMBER, METHOD FOR PRODUCING INTERMEDIATE TRANSFER MEMBER, AND IMAGE FORMING APPARATUS Konica Minolta, Inc. (JP) 2018-05-17 US disclosed
US-20180136590-A1 INTERMEDIATE TRANSFER MEMBER, METHOD FOR PRODUCING INTERMEDIATE TRANSFER MEMBER, AND IMAGE FORMING APPARATUS Konica Minolta, Inc. (JP) 2018-05-17 US disclosed
US-6166013-A Glucocortiocoid-selective agents ABBOTT LABORATORIES (US) 2000-12-26 US disclosed