Morpholine

Morpholine

SCHEMBL6559574

C1COCCN1.CC#N.O=S(=O)(O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Morpholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
CYP2C9 P11712 1/20 0.46
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
GABRA1 P14867 1/20 0.32
TSHR P16473 1/20 0.32
GABRG2 P18507 1/20 0.32
NFKB1 P19838 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRA6 Q16445 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL27791864 0.91 MEN1 (0.50) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL6686007 0.90 MEN1 (0.41) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL1508329 0.88 MEN1 (0.39) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL546382 0.86
Morpholine SCHEMBL2808231 0.86 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL2808233 0.86 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL28072685 0.86 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL7100628 0.84 MEN1 (0.58) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL15789448 0.84 MEN1 (0.58) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL15789446 0.84 MEN1 (0.58) MEN1KMT2AKDM4EGAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6764613-B2 FOR USE IN BLEACHING AND CLEANING MID-AMERICA COMMERCIALIZATION CORPORATION 2004-07-20 US claimed
EP-1036070-B1 N-ALKYL AMMONIUM ACETONITRILE SALTS, METHODS THEREFOR AND COMPOSITIONS THEREWITH CLOROX CO (US) 2004-02-18 EP claimed
US-20030080319-A1 N-alkyl ammonium acetonitrile salts, methods therefor and compositions therewith THE CLOROX COMPANY 2003-05-01 US claimed
EP-1036070-A4 N-ALKYL AMMONIUM ACETONITRILE SALTS, METHODS THEREFOR AND COMPOSITIONS THEREWITH CLOROX CO (US) 2001-01-31 EP claimed
EP-1036070-A1 N-ALKYL AMMONIUM ACETONITRILE SALTS, METHODS THEREFOR AND COMPOSITIONS THEREWITH The Clorox Company (US) 2000-09-20 EP claimed
WO-1998023602-A1 N-ALKYL AMMONIUM ACETONITRILE SALTS, METHODS THEREFOR AND COMPOSITIONS THEREWITH THE CLOROX COMPANY (US) 1998-06-04 WO claimed
US-20040067863-A1 Enclosed bleach activators SPECKMANN HORST-DIETER (DE) 2004-04-08 US disclosed
US-6407045-B1 CLEANING DISHES BY FORMING AQUEOUS CLEANING SOLUTION WITH A SOLID DETERGENT; CONTACTING A DISH SURFACE IN NEED OF CLEANING WITH A CLEANING- EFFECTIVE AMOUNT OF THE CLEANING SOLUTION HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2002-06-18 US disclosed
US-20020032139-A1 Particulate acetonitrile derivatives as bleach activators in solid detergents NITSCH CHRISTIAN (DE) 2002-03-14 US disclosed