Morpholine

Morpholine

SCHEMBL1508329

C1COCCN1.CC#N.COS(=O)(=O)O

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of Morpholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL9984285 0.90 MEN1 (0.48) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL6559574 0.88 MEN1 (0.46) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL6686007 0.83 MEN1 (0.41) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL27288614 0.81 MEN1 (0.39) MEN1KMT2AKDM4EGAACYP2C9
Piperidine SCHEMBL8407029 0.81 ALDH1A1 (0.36)
Morpholine SCHEMBL27791864 0.80 MEN1 (0.50) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL546382 0.79
Morpholine SCHEMBL7100628 0.77 MEN1 (0.58) MEN1KMT2AKDM4EGAACYP2C9
Acetonitrile SCHEMBL1470516 0.77 SLC6A2 (0.30)
Acetonitrile SCHEMBL5157906 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261686-B1 MULTIPHASE MOULDED DETERGENT BODIES WITH NON-PRESSED PARTS HENKEL AG & CO KGAA (DE) 2016-06-15 EP claimed
EP-1141191-A1 PHOSPHATE COMPOUNDS Henkel Kommanditgesellschaft auf Aktien (DE) 2001-10-10 EP claimed
US-6211130-B1 Use of quaternary acetonitrile compounds as activators for detergents HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2001-04-03 US claimed
EP-1045894-A1 DISH WASHING DETERGENT SHAPED BODY WITH SPECIFIC VOLUMETRIC PROPORTIONS Henkel Kommanditgesellschaft auf Aktien (DE) 2000-10-25 EP claimed
EP-1045895-A1 SPECIFIC SHAPED MOULDED BODY DISHWASHER DETERGENTS Henkel Kommanditgesellschaft auf Aktien (DE) 2000-10-25 EP claimed
EP-1044256-A1 METHOD FOR PRODUCING A DISH WASHING DETERGENT SHAPED BODY Henkel Kommanditgesellschaft auf Aktien (DE) 2000-10-18 EP claimed
WO-2000060046-A1 DETERGENTS FOR DISHWASHING MACHINE WITH PARTICLE-TYPE CLEAR-RINSING AGENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-10-12 WO claimed
WO-2000039260-A1 PHOSPHATE COMPOUNDS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-07-06 WO claimed
WO-1999035233-A1 METHOD FOR PRODUCING A DISH WASHING DETERGENT SHAPED BODY HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-07-15 WO claimed
WO-1999035232-A1 DISH WASHING DETERGENT SHAPED BODY WITH SPECIFIC VOLUMETRIC PROPORTIONS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-07-15 WO claimed
WO-1999035236-A1 SPECIFIC SHAPED MOULDED BODY DISHWASHER DETERGENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-07-15 WO claimed
EP-2864463-A1 DISHWASHING DETERGENT Henkel AG&Co. KGAA (DE) 2015-04-29 EP disclosed
WO-2013182510-A1 DISHWASHING DETERGENT HENKEL AG & CO. KGAA (DE) 2013-12-12 WO disclosed
EP-2294172-A1 BACITRACIN METAL COMPLEXES USED AS BLEACH CATALYSTS Henkel AG & Co. KGaA (DE) 2011-03-16 EP disclosed
WO-2009150009-A1 BACITRACIN METAL COMPLEXES USED AS BLEACH CATALYSTS HENKEL AG & CO. KGAA (DE) 2009-12-17 WO disclosed
WO-1998023533-A1 LIQUID COMPOSITIONS CONTAINING N-ALKYL AMMONIUM ACETONITRILE SALTS THE CLOROX COMPANY (US) 1998-06-04 WO disclosed
US-5741437-A SOURCE OF ACTIVE OXYGEN REACTS WITH NITRILE FOR BLEACHING APPLICATIONS THE CLOROX COMPANY (US) 1998-04-21 US disclosed
US-5739327-A OXYGEN BLEACHES OF NITRILE BONDED TO QUATERNARY NITROGEN THE CLOROX COMPANY (US) 1998-04-14 US disclosed
EP-0775127-A1 N-ALKYL AMMONIUM ACETONITRILE BLEACH ACTIVATORS The Clorox Company (US) 1997-05-28 EP disclosed
WO-1996040661-A1 N-ALKYL AMMONIUM ACETONITRILE BLEACH ACTIVATORS THE CLOROX COMPANY (US) 1996-12-19 WO disclosed