SCHEMBL6559997

SCHEMBL6559997

CCCc1cc(=O)oc2c(CCC)c(O)ccc12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 9/20 0.71
KDM4E B2RXH2 8/20 0.71
GLA P06280 8/20 0.71
ALDH1A1 P00352 8/20 0.71
HPGD P15428 6/20 0.71
HIF1A Q16665 4/20 0.71
ERAP1 Q9NZ08 6/20 0.70
KMT2A Q03164 3/20 0.70
POLB P06746 1/20 0.70
CYP1A2 P05177 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C19 P33261 1/20 0.68
MEN1 O00255 2/20 0.67
CASP1 P29466 1/20 0.67
CASP7 P55210 1/20 0.67
HSD17B10 Q99714 1/20 0.67
USP2 O75604 1/20 0.61
HSD17B3 P37058 1/20 0.57
ATM Q13315 1/20 0.56
MCL1 Q07820 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560136 0.94 KDM4E (0.64) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL14756049 0.93 GAA (0.70) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL15211319 0.90 MCL1 (0.66) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL6561714 0.88 KDM4E (0.58) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL15295521 0.87 MCL1 (0.70) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL15984890 0.85 KDM4E (0.64) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL11079352 0.85 GAA (0.63) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL15082524 0.84 GAA (0.62) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL31454860 0.83 ALDH1A1 (0.58) GAAKDM4EGLAALDH1A1HPGD
SCHEMBL17615425 0.82 ERN1 (0.66) GAAKDM4EGLAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed