SCHEMBL6560136

SCHEMBL6560136

CCCc1c(O)ccc2c(CC)cc(=O)oc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.64
ALDH1A1 P00352 7/20 0.64
GAA P10253 6/20 0.64
HPGD P15428 6/20 0.64
GLA P06280 6/20 0.64
HIF1A Q16665 2/20 0.64
ERAP1 Q9NZ08 5/20 0.63
KMT2A Q03164 3/20 0.63
MEN1 O00255 2/20 0.63
ATM Q13315 1/20 0.63
CASP1 P29466 1/20 0.63
CASP7 P55210 1/20 0.63
HSD17B10 Q99714 1/20 0.63
POLB P06746 1/20 0.62
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C19 P33261 1/20 0.61
USP2 O75604 1/20 0.56
MCL1 Q07820 2/20 0.52
MAOB P27338 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559997 0.94 GAA (0.71) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL15211319 0.90 MCL1 (0.66) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL14756049 0.90 GAA (0.70) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6561714 0.88 KDM4E (0.58) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL11079352 0.85 GAA (0.63) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL13836162 0.84 ALDH1A1 (0.55) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6561597 0.82 ALDH1A1 (0.51) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL14898335 0.81 MCL1 (0.77) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL1594333 0.81 CSNK2A2 (0.61) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL15295521 0.81 MCL1 (0.70) KDM4EALDH1A1GAAHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed