SCHEMBL6561714

SCHEMBL6561714

CCCc1c(O)ccc2c(CC(C)(C)C)cc(=O)oc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
GAA P10253 6/20 0.58
ALDH1A1 P00352 6/20 0.58
GLA P06280 6/20 0.58
HPGD P15428 6/20 0.58
HIF1A Q16665 2/20 0.58
KMT2A Q03164 4/20 0.57
MEN1 O00255 2/20 0.57
CASP1 P29466 2/20 0.57
CASP7 P55210 2/20 0.57
HSD17B10 Q99714 2/20 0.57
ERAP1 Q9NZ08 6/20 0.57
POLB P06746 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C19 P33261 1/20 0.56
ATM Q13315 1/20 0.51
USP2 O75604 1/20 0.51
MCL1 Q07820 2/20 0.47
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560136 0.88 KDM4E (0.64) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL6559997 0.88 GAA (0.71) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL15211319 0.84 MCL1 (0.66) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL6561597 0.82 ALDH1A1 (0.51) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL14756049 0.81 GAA (0.70) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL11079352 0.80 GAA (0.63) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL5205948 0.79 KDM4E (0.37) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL1594333 0.78 CSNK2A2 (0.61) KDM4EGAAALDH1A1GLAHPGD
SCHEMBL6559981 0.76 PDE5A (0.48) KDM4EALDH1A1HPGDKMT2APOLB
SCHEMBL15295521 0.75 MCL1 (0.70) KDM4EGAAALDH1A1GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed