SCHEMBL6560048

SCHEMBL6560048

COc1ccc(C2CC(C(F)(F)F)=NN2c2ccc(S(N)(=O)=O)cc2)c(F)c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.60
PTGS2 P35354 4/20 0.60
CA1 P00915 8/20 0.58
CA2 P00918 8/20 0.58
ACHE P22303 6/20 0.58
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230657 0.90 CA2 (0.71) PTGS1PTGS2CA1CA2ACHE
SCHEMBL5858805 0.90 PTGS1 (0.60) PTGS1PTGS2CA1CA2ACHE
SCHEMBL5857642 0.87 PTGS1 (0.63) PTGS1PTGS2
Enflicoxib SCHEMBL26427 0.86 PTGS1 (0.66) PTGS1PTGS2CA1CA2ACHE
SCHEMBL5857924 0.85 PTGS1 (0.64) PTGS1PTGS2CA2
SCHEMBL5858890 0.85 PTGS1 (0.63) PTGS1PTGS2
SCHEMBL5856299 0.84 L3MBTL1 (0.71) PTGS1PTGS2CA1CA2L3MBTL1
SCHEMBL5857443 0.84 CA2 (0.64) PTGS1PTGS2CA1CA2ACHE
SCHEMBL5856805 0.82 PTGS1 (0.74) PTGS1PTGS2
SCHEMBL5856591 0.81 PTGS1 (0.67) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083171-B1 PYRAZOLINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-04-28 EP claimed