SCHEMBL6560672

SCHEMBL6560672

CNC(=O)C=C(Cc1ccc(OC)cc1)c1cccc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.52
APBA1 Q02410 1/20 0.52
PTPN1 P18031 1/20 0.47
ALDH1A1 P00352 3/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
KDM4E B2RXH2 1/20 0.47
DRD4 P21917 1/20 0.47
MTNR1A P48039 1/20 0.46
GCGR P47871 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.45
PLK1 P53350 1/20 0.45
NPC1 O15118 2/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.43
MCL1 Q07820 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561772 0.87 POLB (0.44) CACNA1BAPBA1PTPN1ALDH1A1KMT2A
SCHEMBL6560700 0.84 NPC1 (0.51) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL6561900 0.80 NPC1 (0.51) CACNA1BAPBA1ALDH1A1KMT2AMEN1
SCHEMBL6560669 0.80 NPC1 (0.51) CACNA1BAPBA1ALDH1A1KMT2AMEN1
SCHEMBL16162267 0.79 TP53 (0.67) CACNA1BAPBA1PTPN1ALDH1A1KMT2A
SCHEMBL6561872 0.74 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL9856912 0.71 GCGR (0.67) CACNA1BAPBA1ALDH1A1KMT2AMTNR1A
SCHEMBL27773350 0.71 CACNA1B (0.50) CACNA1BAPBA1PTPN1ALDH1A1KMT2A
SCHEMBL16162265 0.69 POLB (0.63) PTPN1ALDH1A1KMT2AMEN1KDM4E
SCHEMBL28813458 0.69 CACNA1B (0.59) CACNA1BAPBA1ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed