SCHEMBL6561061

SCHEMBL6561061

CC1(C)C=Cc2cc(N)ccc21

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
CASP1 P29466 2/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
PDE10A Q9Y233 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18989196 0.75 HTR2C (0.36) CA12CA2CA9
SCHEMBL23190235 0.75 HTR2C (0.36) ALDH1A1CYP3A4TSHR
SCHEMBL29387054 0.69 KDM4E (0.39) PDK2
SCHEMBL23671508 0.67 MAPT (0.35) ALDH1A1
Ammonia Solution, Strong SCHEMBL7086115 0.67 KDM4E (0.38) PDK2
SCHEMBL28056042 0.67 KDM4E (0.38) PDK2
SCHEMBL27414073 0.67 KDM4E (0.38) PDK2
SCHEMBL2012004 0.67 HIF1A (0.46) ALDH1A1CA12CA1CA2CA9
SCHEMBL29647889 0.67 ALDH1A1 (0.38) ALDH1A1CASP1CYP3A4TSHRPDE10A
SCHEMBL8970935 0.67 ALDH1A1 (0.38) ALDH1A1CASP1CYP3A4TSHRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1085009-B1 INDAN DERIVATIVES NISSAN CHEMICAL IND LTD (JP) 2004-11-10 EP disclosed
US-6486178-B1 Indane derivatives NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2002-11-26 US disclosed
EP-1085009-A1 INDAN DERIVATIVES Nissan Chemical Industries, Ltd. (JP) 2001-03-21 EP disclosed
WO-1994014801-A1 HETEROCYCLIC UREA DERIVATIVES AS 5HT2C AND 5HT2B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed