SCHEMBL2012004

SCHEMBL2012004

CC1(C)C=Cc2cc(N)ccc2O1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 11/20 0.46
EPAS1 Q99814 11/20 0.46
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA9 Q16790 2/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
CA7 P43166 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CA13 Q8N1Q1 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP3A4 P08684 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL4801415 0.91 ALDH1A1 (0.48) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL3193312 0.85 ODC1 (0.47) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL4800628 0.80 PTGS1 (0.53) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL3049240 0.79 ALDH1A1 (0.46) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL7738844 0.79 HIF1A (0.58) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL28405015 0.79 HIF1A (0.50) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL9219622 0.78 HTR2C (0.54) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL30140565 0.78 XDH (0.68) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL6024450 0.78 HTR2C (0.54) HIF1AEPAS1ALDH1A1HPGDCA12
SCHEMBL8723354 0.78 XDH (0.68) HIF1AEPAS1ALDH1A1HPGDCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160168161-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND NISSAN CHEMICAL INDUSTIES, LTD. (JP) 2016-06-16 US claimed
EP-3026047-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND Nissan Chemical Industries, Ltd. (JP) 2016-06-01 EP claimed
CN-105377826-A Process for producing heterocyclic compound NISSAN CHEMICAL IND LTD 2016-03-02 CN claimed
EP-1535918-B1 PROCESS FOR PRODUCING AMINOBENZOPYRAN COMPOUND NISSAN CHEMICAL IND LTD (JP) 2010-11-03 EP claimed
US-7683189-B2 Process for producing aminobenzopyran compound NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2010-03-23 US claimed
US-20050192444-A1 Process for producing aminobenzopyran compound NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2005-09-01 US claimed
EP-1535918-A1 PROCESS FOR PRODUCING AMINOBENZOPYRAN COMPOUND Nissan Chemical Industries, Ltd. (JP) 2005-06-01 EP claimed
CN-109096235-B 2, 2-dimethyl benzopyran derivative and preparation method and application thereof 沈阳药科大学 2022-06-21 CN disclosed
US-20160168161-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND NISSAN CHEMICAL INDUSTIES, LTD. (JP) 2016-06-16 US disclosed
US-20160168161-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND NISSAN CHEMICAL INDUSTIES, LTD. (JP) 2016-06-16 US disclosed
US-20160168161-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND NISSAN CHEMICAL INDUSTIES, LTD. (JP) 2016-06-16 US disclosed
EP-3026047-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND Nissan Chemical Industries, Ltd. (JP) 2016-06-01 EP disclosed
CN-105377826-A Process for producing heterocyclic compound NISSAN CHEMICAL IND LTD 2016-03-02 CN disclosed
WO-2005090357-A1 TRICYCLIC BENZOPYRAN COMPOUND AS ANTI-ARRHYTHMIC AGENTS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2005-09-29 WO disclosed
US-20050203145-A1 6-alkylamino-2,2'-disubstituted-7,8-disubstituted-2H-1-benzopyran derivatives as 5-lipoxygenase inhibitor KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY 2005-09-15 US disclosed
US-20050192444-A1 Process for producing aminobenzopyran compound NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2005-09-01 US disclosed
EP-1535918-A1 PROCESS FOR PRODUCING AMINOBENZOPYRAN COMPOUND Nissan Chemical Industries, Ltd. (JP) 2005-06-01 EP disclosed
US-5416097-A Potassium channel activators/openers BERLEX LABORATORIES, INC. (US) 1995-05-16 US disclosed
US-5164509-A BENZODIAZOLO ANALOGS E. R. SQUIBB & SONS, INC. (US) 1992-11-17 US disclosed
EP-0488107-A2 Tricyclic benzodiazole analogs and their use in the treatment of cardiovascular disorders E.R. SQUIBB & SONS, INC. (US) 1992-06-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050192444-A1 Process for producing aminobenzopyran compound ALDH7A1, ACMSD, MANBA HIF1A 404/4885EPAS1 3320/4885ALDH1A1 195/4885
US-20160168161-A1 METHOD FOR PRODUCING HETEROCYCLIC COMPOUND H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NAT1, NAT10 HIF1A 3098/4885EPAS1 4052/4885ALDH1A1 2486/4885
US-20050203145-A1 6-alkylamino-2,2'-disubstituted-7,8-disubstituted-2H-1-benzopyran derivatives as 5-lipoxygenase inhibitor ALOX5, LOX, ALOX15 HIF1A 1100/4885EPAS1 1588/4885ALDH1A1 1656/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.