SCHEMBL6561366

SCHEMBL6561366

CCOc1nc2ccccc2nc1NC(=O)Oc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
LMNA P02545 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
FAAH O00519 6/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560382 0.85 ALDH1A1 (0.50) KDM4ELMNAMEN1KMT2AALDH1A1
SCHEMBL7803121 0.82 MAPT (0.43) MEN1KMT2AMAPTGAA
SCHEMBL7803067 0.82 MAPT (0.51) HSD17B10MEN1KMT2AMAPTGAA
SCHEMBL7804711 0.81 MAPT (0.43) KDM4ELMNAKMT2ARAB9AALDH1A1
SCHEMBL7800966 0.80 NPC1 (0.51) KDM4ELMNAMEN1KMT2ARAB9A
SCHEMBL7803529 0.79 CCKAR (0.43) KDM4ELMNAMEN1KMT2AALDH1A1
SCHEMBL27456552 0.74 ALDH1A1 (0.54) MEN1KMT2AFAAHRAB9AALDH1A1
SCHEMBL6560060 0.74 RAB9A (0.47) KDM4ELMNAMEN1KMT2AFAAH
SCHEMBL8380443 0.73 KDM4E (0.59) KDM4ELMNAHSD17B10MEN1KMT2A
SCHEMBL8699761 0.73 RAB9A (0.43) KDM4EKMT2AFAAHRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075469-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2004-05-26 EP disclosed
US-6683184-B2 ANTITUMOR AGENTS SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2004-01-27 US disclosed
US-20030092910-A1 Piperazine derivatives and process for the preparation thereof SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2003-05-15 US disclosed
EP-1075469-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2001-02-14 EP disclosed
WO-2000052001-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030092910-A1 Piperazine derivatives and process for the preparation thereof CBR1, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HCCS KDM4E 2023/4885LMNA 3343/4885HSD17B10 1124/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.