SCHEMBL6561440

SCHEMBL6561440

CC1CCC2C(N)=Nc3cc(NCc4cccc(Cl)c4)ccc3C12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.53
NOS3 P29474 7/20 0.53
NOS1 P29475 7/20 0.53
CCNT1 O60563 3/20 0.40
CDK9 P50750 3/20 0.40
MAOB P27338 2/20 0.37
HTR6 P50406 1/20 0.37
APP P05067 2/20 0.37
HRH4 Q9H3N8 1/20 0.37
RAF1 P04049 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6069708 0.76 NTRK1 (0.41) NOS2NOS3NOS1CCNT1CDK9
Hydrochloric Acid SCHEMBL6069850 0.73 NOS3 (0.52) NOS2NOS3NOS1MAOBHTR6
SCHEMBL6069550 0.71 NOS3 (0.39) NOS2NOS3NOS1
SCHEMBL6561433 0.70 NOS1 (0.98) NOS2NOS3NOS1
Hydrochloric Acid SCHEMBL6069807 0.70 NOS1 (1.00) NOS2NOS3NOS1
SCHEMBL6561322 0.68 NOS1 (0.69) NOS2NOS3NOS1
Hydrochloric Acid SCHEMBL6069274 0.67 NOS1 (0.71) NOS2NOS3NOS1
SCHEMBL6561325 0.67 NOS1 (0.98) NOS2NOS3NOS1
SCHEMBL6700054 0.66 CHRM2 (0.55) MAOBHTR6APP
SCHEMBL632217 0.66 CHRM2 (0.55) MAOBHTR6APPMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115708-B1 AMINOALKYL-3,4-DIHYDROQUINOLINE DERIVATES AS NO-SYNTHASE INHIBITORS SCHERING AG (DE) 2004-04-14 EP claimed