Flavone

Flavone

SCHEMBL6561748

O=C(O)[C@H]1OC(O)[C@H](O)[C@@H](O)[C@@H]1O.O=c1cc(-c2ccccc2)oc2ccccc12

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 10/20 0.62
GABRP O00591 4/20 0.62
GABRD O14764 4/20 0.62
GABRA1 P14867 4/20 0.62
GABRB1 P18505 4/20 0.62
GABRG2 P18507 4/20 0.62
GABRB3 P28472 4/20 0.62
GABRA5 P31644 4/20 0.62
GABRA3 P34903 4/20 0.62
GABRA2 P47869 4/20 0.62
GABRB2 P47870 4/20 0.62
GABRA4 P48169 4/20 0.62
GABRE P78334 4/20 0.62
GABRA6 Q16445 4/20 0.62
GABRG1 Q8N1C3 4/20 0.62
GABRG3 Q99928 4/20 0.62
GABRQ Q9UN88 4/20 0.62
PARP1 P09874 4/20 0.62
TNKS2 Q9H2K2 4/20 0.62
HPGD P15428 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flavone SCHEMBL21823959 1.00 TNKS (0.62) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL28655692 0.83 TNKS (0.62) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL29013778 0.83 TNKS (0.62) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL344911 0.83 TNKS (0.62) TNKSGABRPGABRDGABRA1GABRB1
Baicalein SCHEMBL28870586 0.81 ABCB1 (0.68) GABRPGABRDGABRA1GABRB1GABRG2
Flavone SCHEMBL31316377 0.79 TNKS (1.00) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL30542161 0.79 TNKS (1.00) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL18879 0.79 TNKS (1.00) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL15676601 0.79 TNKS (1.00) TNKSGABRPGABRDGABRA1GABRB1
Flavone SCHEMBL28248986 0.79 TNKS (1.00) TNKSGABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114807082-A Liverwort flavonoid glucuronic acid glycosyl transferase and coding gene and application thereof 山东大学 2022-07-29 CN claimed
CN-106606507-B Application of flavone diglucuronide compound in preparation of cyclooxygenase inhibitor 上海医药工业研究院 2021-06-25 CN claimed
CN-104800414-B The separation method of general flavone glucuronide and total benzyl carbinol glycosides in callicarpa kwangtungensis Chun 江苏康缘药业股份有限公司 2019-03-26 CN claimed
WO-2015019381-A1 METHOD FOR IN VITRO DIAGNOSIS OF IDIOPATHIC PULMONARY FIBROSIS SALTINI CESARE (IT) 2015-02-12 WO claimed
CN-114807082-A Liverwort flavonoid glucuronic acid glycosyl transferase and coding gene and application thereof 山东大学 2022-07-29 CN disclosed
US-20220143058-A1 Pharmaceutical Compositions Comprising a Hydroxyethylquercetin Glucuronide JANSSEN PHARMACEUTICA NV (BE) 2022-05-12 US disclosed
CN-114432323-A Application of flavonoid compound in preparation of medicine for preventing or treating acute lung injury and/or acute respiratory distress syndrome 苏州凯祥生物科技有限公司 2022-05-06 CN disclosed
EP-3860617-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING A HYDROXYETHYLQUERCETIN GLUCURONIDE Janssen Pharmaceutica N.V. (BE) 2021-08-11 EP disclosed
CN-106606507-B Application of flavone diglucuronide compound in preparation of cyclooxygenase inhibitor 上海医药工业研究院 2021-06-25 CN disclosed
US-20200155584-A1 Pharmaceutical Compositions Comprising a Hydroxyethylquercetin Glucuronide JANSSEN PHARMACEUTICA NV (BE) 2020-05-21 US disclosed
US-10639294-B2 Pharmaceutical compositions comprising a hydroxyethylquercetin glucuronide metabolite JANSSEN PHARMACEUTICA NV (BE) 2020-05-05 US disclosed
WO-2020070643-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING A HYDROXYETHYLQUERCETIN GLUCURONIDE JANSSEN PHARMACEUTICA NV (BE) 2020-04-09 WO disclosed
CN-104800414-B The separation method of general flavone glucuronide and total benzyl carbinol glycosides in callicarpa kwangtungensis Chun 江苏康缘药业股份有限公司 2019-03-26 CN disclosed
US-20160339070-A1 USE OF HERBAL SAPONINS TO REGULATE GUT MICROFLORA HSIAO, WEN LUAN WENDY (HK) 2016-11-24 US disclosed
US-20150126463-A1 USE OF HERBAL SAPONINS TO REGULATE GUT MICROFLORA HONG KONG BAPTIST UNIVERSITY (HK) 2015-05-07 US disclosed
WO-2015062556-A1 USE OF HERBAL SAPONINS TO REGULATE GUT MICROFLORA HONG KONG BAPTIST UNIVERSITY (CN) 2015-05-07 WO disclosed
WO-2015019381-A1 METHOD FOR IN VITRO DIAGNOSIS OF IDIOPATHIC PULMONARY FIBROSIS SALTINI CESARE (IT) 2015-02-12 WO disclosed
EP-1397502-A2 DNA SEQUENCING OF ABC TRANSPORTER OR MULTI DRUG RESISTANT PROTEIN FOR BETTER ENVIRONMENT STRESS TOLERANT CROPS Avestha Gengraine Technologies PVT Ltd (IN) 2004-03-17 EP disclosed
WO-2002083911-A1 PRODUCTION OF PLANTS WITH INCREASED TOLERANCE TO DROUGHT STRESS OR WITH INCREASED TRANSPIRATION MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2002-10-24 WO disclosed
WO-2002057406-A2 DNA SEQUENCING OF ABC TRANSPORTER OR MULTI DRUG RESISTANT PROTEIN FOR BETTER ENVIRONMENT STRESS TOLERANT CROPS AVESTHA GENGRAINE TECHNOLOGIES PVT LTD (IN) 2002-07-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220143058-A1 Pharmaceutical Compositions Comprising a Hydroxyethylquercetin Glucuronide COMT, UGT1A6, SLC6A2 TNKS 4314/4885GABRP 753/4885GABRD 593/4885
US-10639294-B2 Pharmaceutical compositions comprising a hydroxyethylquercetin glucuronide metabolite UGT1A7, COMT, UGT1A6 TNKS 4216/4885GABRP 1114/4885GABRD 628/4885
US-20200155584-A1 Pharmaceutical Compositions Comprising a Hydroxyethylquercetin Glucuronide COMT, UGT1A6, SLC6A2 TNKS 4314/4885GABRP 753/4885GABRD 593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.