SCHEMBL6561848

SCHEMBL6561848

Cc1cc(C#CCNc2ccc(C(=N)N)cc2)ccc1C(=O)N1CCC(N)C1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 15/20 0.41
F2 P00734 1/20 0.39
PLG P00747 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
ST14 Q9Y5Y6 1/20 0.39
ACACB O00763 1/20 0.37
CDK1 P06493 1/20 0.37
PIK3CA P42336 2/20 0.37
MTOR P42345 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561958 0.87 ACACB (0.49) F2PLGPRSS1PRSS2PRSS3
SCHEMBL6561944 0.84 F10 (0.43) ACACBPIK3CAMTOR
SCHEMBL6565512 0.83 GAA (0.40) F2PRSS1ACACB
SCHEMBL6565424 0.80 ITGB3 (0.42) F2PRSS1
SCHEMBL6562282 0.80 PIK3CA (0.44) F2PLGACACBPIK3CAMTOR
SCHEMBL6564957 0.78 F2 (0.38) F2PRSS1
SCHEMBL6565351 0.78 F10 (0.44) F2PLGPRSS1PRSS2PRSS3
SCHEMBL5885702 0.78 ACACB (0.46) PRSS1ACACB
SCHEMBL6563137 0.77 KLK5 (0.37) F2PLGPRSS1PRSS2PRSS3
Hydrochloric Acid SCHEMBL5886024 0.77 ACACB (0.46) PRSS1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed