SCHEMBL6561961

SCHEMBL6561961

Cc1ccc(C(=O)N(C)CCc2ccccc2)cc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.39
CTSK P43235 3/20 0.38
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
PTGES O14684 1/20 0.34
NPY5R Q15761 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPK14 Q16539 1/20 0.34
CTSS P25774 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
NAMPT P43490 1/20 0.33
PTPN11 Q06124 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565333 0.92 MEN1 (0.40) PTGESCTSSCTSLCTSBACACB
SCHEMBL6563537 0.88 PLAU (0.38) PTGESNPC1RAB9APTPN11ACACB
SCHEMBL6563455 0.85 RAB9A (0.41) CTSKNPC1RAB9ANAMPTESRRG
SCHEMBL6561959 0.85 MLYCD (0.41) MLYCDROCK2ROCK1TLR9TLR8
SCHEMBL6565428 0.82 MEN1 (0.34) NPC1RAB9APTPN11ACACB
SCHEMBL6563229 0.82 PLAU (0.37) PTGESNPC1RAB9APTPN11ACACB
SCHEMBL6565278 0.81 PTPN11 (0.33) PTPN11
SCHEMBL6565492 0.80 CNR2 (0.39) NPC1RAB9APTPN11ACACBABL1
SCHEMBL6563932 0.80 HTT (0.34) PTGESNPC1RAB9APTPN11ACACB
SCHEMBL6565352 0.80 PTPN11 (0.33) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed