SCHEMBL6565333

SCHEMBL6565333

Cc1ccc(C(=O)N(C)Cc2ccccc2)cc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
PTGES O14684 1/20 0.39
HTT P42858 1/20 0.38
LIMK2 P53671 6/20 0.38
LMNA P02545 1/20 0.38
ADORA2A P29274 1/20 0.37
HPGD P15428 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
LIMK1 P53667 2/20 0.36
ACACB O00763 1/20 0.36
ABL1 P00519 1/20 0.36
LCK P06239 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561961 0.92 MLYCD (0.39) CTSLCTSBCTSSPTGESLMNA
SCHEMBL6563537 0.89 PLAU (0.38) KMT2APTGESHTTTSHRACACB
SCHEMBL6561871 0.84 KMT2A (0.46) MEN1KMT2AHTTLIMK2ADORA2A
SCHEMBL6565428 0.84 MEN1 (0.34) MEN1KMT2AALDH1A1GAATSHR
SCHEMBL6563455 0.83 RAB9A (0.41) LMNASMN1; SMN2
SCHEMBL6563229 0.83 PLAU (0.37) KMT2APTGESHTTALDH1A1TSHR
SCHEMBL6563932 0.82 HTT (0.34) MEN1KMT2APTGESHTTTSHR
SCHEMBL6565492 0.82 CNR2 (0.39) MEN1KMT2AHPGDALDH1A1GAA
SCHEMBL6565352 0.81 PTPN11 (0.33)
SCHEMBL6565278 0.80 PTPN11 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed