SCHEMBL6562815

SCHEMBL6562815

O=C(O)c1ccc(-c2cccc(O)c2)nc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.70
HSD17B1 P14061 3/20 0.63
HSD17B2 P37059 3/20 0.63
CHEK1 O14757 1/20 0.62
P4HA1 P13674 2/20 0.59
P4HTM Q9NXG6 1/20 0.59
HPGDS O60760 1/20 0.52
CYP4F2 P78329 1/20 0.50
CYP4A11 Q02928 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA6 P23280 1/20 0.50
CA9 Q16790 1/20 0.50
KDM1A O60341 1/20 0.50
BAZ2B Q9UIF8 1/20 0.49
METAP2 P50579 1/20 0.49
AKR1C3 P42330 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL503140 0.90 LDHA (0.79) LDHAHSD17B1HSD17B2CHEK1P4HA1
SCHEMBL31243316 0.88 LDHA (0.77) LDHAHSD17B1HSD17B2CHEK1P4HA1
SCHEMBL1785610 0.86 HPGDS (0.71) LDHAHSD17B1HSD17B2CHEK1HPGDS
SCHEMBL505455 0.83 LDHA (1.00) LDHAP4HA1P4HTMHPGDSBAZ2B
SCHEMBL2560542 0.83 LDHA (0.68) LDHAHSD17B1HSD17B2P4HA1P4HTM
SCHEMBL1543156 0.83 HPGDS (0.76) LDHAP4HA1P4HTMHPGDSCYP4F2
SCHEMBL21228142 0.82 HSD17B1 (0.56) LDHAHSD17B1HSD17B2CHEK1HPGDS
SCHEMBL29914699 0.82 HSD17B1 (0.56) LDHAHSD17B1HSD17B2CHEK1HPGDS
SCHEMBL3226145 0.81 CHEK1 (0.55) LDHAHSD17B1HSD17B2CHEK1HPGDS
SCHEMBL9939612 0.81 LDHA (0.57) LDHAHSD17B1HSD17B2CHEK1P4HA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019149205-A1 BENZOHETEROARYL DERIVATIVE AND PREPARATION METHOD AND MEDICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2019-08-08 WO disclosed
EP-2142516-B1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS SANOFI SA (FR) 2012-12-26 EP disclosed
EP-1235777-B1 VITAMIN D ANALOGUES GALDERMA RES & DEV (FR) 2004-06-16 EP disclosed
EP-1235777-A2 VITAMIN D ANALOGUES Galderma Research & Development, S.N.C. (FR) 2002-09-04 EP disclosed
WO-2001038303-A2 VITAMIN D ANALOGUES GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2001-05-31 WO disclosed