SCHEMBL6562867

SCHEMBL6562867

CC(CNS(=O)(=O)C(C)C)c1ccc(CCNC(=O)OCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 9/20 0.55
GRIA2 P42262 1/20 0.51
CA5A P35218 2/20 0.50
CA2 P00918 1/20 0.50
MAPT P10636 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTT P42858 1/20 0.44
CA1 P00915 2/20 0.44
CA4 P22748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561724 0.94 GRIA4 (0.51) GRIA4GRIA2CA5ACA2MAPT
SCHEMBL6563108 0.91 CA1 (0.50) GRIA4GRIA2CA5ACA2MAPT
SCHEMBL5877953 0.81 GRIA4 (0.64) GRIA4GRIA2CA5ACA2CA1
SCHEMBL5878181 0.80 GRIA4 (0.69) GRIA4GRIA2MAPTL3MBTL1SMN1; SMN2
SCHEMBL5878118 0.79 GRIA4 (0.64) GRIA4GRIA2CA2CA1
SCHEMBL5877766 0.78 GRIA4 (0.72) GRIA4GRIA2SMN1; SMN2
SCHEMBL6563303 0.77 GRIA4 (0.80) GRIA4GRIA2
Benzyl Phenethylcarbamate SCHEMBL4287199 0.77 LMNA (0.73) CA2MAPTL3MBTL1LMNASMN1; SMN2
SCHEMBL205765 0.77 MGLL (0.65) MAPTL3MBTL1LMNASMN1; SMN2HTT
SCHEMBL5877621 0.77 GRIA4 (0.70) GRIA4GRIA2CA2CA1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296945-B1 SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6703425-B2 ADMINISTERING GLUTAMATE RECEPTOR POTENTIATOR TO TREAT PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY 2004-03-09 US disclosed
US-20030229102-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-11 US disclosed
EP-1296945-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2003-04-02 EP disclosed
WO-2001096289-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229102-A1 Sulfonamide derivatives GRIN1, GRIN2A, SLC1A2 GRIA4 17/4885GRIA2 8/4885CA5A 1275/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.