SCHEMBL6563265

SCHEMBL6563265

Cc1ccc(C#CCNc2ccc(C#N)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
CYP2A6 P11509 2/20 0.55
MAPT P10636 2/20 0.44
CSNK1A1 P48729 1/20 0.39
CSNK1D P48730 1/20 0.39
GSK3B P49841 1/20 0.39
CSNK1G2 P78368 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
KCNH2 Q12809 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
RORC P51449 1/20 0.39
HTT P42858 3/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565480 0.89 GSK3B (0.47) ALDH1A1CYP2A6GSK3BRORCLMNA
SCHEMBL6563318 0.89 BCHE (0.49) ALDH1A1CYP2A6MAPTMEN1KMT2A
SCHEMBL28944597 0.84 GRM5 (0.47) ALDH1A1CYP2A6GSK3BLOXL2GRM5
SCHEMBL6563225 0.83 IDO1 (0.44) ALDH1A1CYP2A6MAPTMEN1KMT2A
SCHEMBL29712697 0.82 MAPT (0.53) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL29712675 0.82 MAPT (0.53) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL6565837 0.82 CYP1A1 (0.44) CSNK1A1CSNK1DGSK3BCSNK1G2GRM5
SCHEMBL6561856 0.79 LMNA (0.47) MAPTCSNK1A1CSNK1DMEN1KMT2A
SCHEMBL11135905 0.78 SMN1; SMN2 (0.52) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL13232516 0.77 MAPT (0.61) ALDH1A1CYP2A6MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed