SCHEMBL6565480

SCHEMBL6565480

Cc1ccc(C(=O)c2ccc(C#CCNc3ccc(C#N)cc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.47
GSK3A P49840 1/20 0.47
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
CYP2A6 P11509 1/20 0.43
VNN1 O95497 4/20 0.40
RORC P51449 2/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
SRD5A2 P31213 1/20 0.39
KCNA5 P22460 1/20 0.39
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563532 0.89 ALDH1A1 (0.44) ALDH1A1LMNAVNN1SMN1; SMN2
SCHEMBL6563265 0.89 ALDH1A1 (0.55) GSK3BALDH1A1LMNACYP2A6RORC
SCHEMBL7670899 0.84 PRSS1 (0.43) ALDH1A1LMNA
SCHEMBL6563651 0.84 MAPK13 (0.45) GSK3BGSK3AALDH1A1SAE1UBA2
SCHEMBL11135905 0.83 SMN1; SMN2 (0.52) ALDH1A1SRD5A2CA1CA2SMN1; SMN2
SCHEMBL6565461 0.82 VNN1 (0.48) LMNAVNN1TDP1
SCHEMBL6563318 0.81 BCHE (0.49) ALDH1A1CYP2A6RORCCA1CA2
SCHEMBL6563777 0.81 GSK3B (0.45) GSK3BALDH1A1SAE1UBA2CA1
SCHEMBL507820 0.81 ALDH1A1 (0.67) GSK3BGSK3AALDH1A1LMNACYP2A6
SCHEMBL6561875 0.80 HPGD (0.47) ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed