SCHEMBL6565016

SCHEMBL6565016

CC(C)CC(OC(=O)NCc1ccccc1)C(=O)N(CC1CCCC(C#N)C1)C1CCNC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 20/20 0.42
SLC6A4 P31645 20/20 0.42
SLC6A3 Q01959 16/20 0.42
CYP2D6 P10635 7/20 0.42
KCNH2 Q12809 6/20 0.41
CHRM4 P08173 1/20 0.37
CYP3A4 P08684 1/20 0.37
CHRM5 P08912 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567334 0.84 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6565786 0.77 CTSS (0.37) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL7021566 0.76 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6563698 0.74 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3
SCHEMBL7434479 0.73 ROCK2 (0.42) SLC6A2SLC6A4SLC6A3
SCHEMBL6565039 0.72 CTSS (0.46)
SCHEMBL7436060 0.72 SLC6A4 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6565014 0.71 CTSL (0.38)
SCHEMBL3894952 0.70 CTSL (0.54)
SCHEMBL7431178 0.69 JAK3 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed