SCHEMBL6565369

SCHEMBL6565369

CCOC(=O)CCC(=O)N(c1cc(C)c(I)cc1C)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
CYP4F2 P78329 2/20 0.33
CYP4A11 Q02928 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CYP1A2 P05177 1/20 0.31
PTPN1 P18031 1/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
PKM P14618 1/20 0.31
KAT2B Q92831 1/20 0.31
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6764579 0.77 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL27623118 0.64 ALDH1A1 (0.48) ALDH1A1MAPTKDM4ECYP1A2PTPN1
SCHEMBL6571937 0.64 ALDH1A1 (0.33) SMN1; SMN2ALDH1A1MAPTKDM4EL3MBTL1
Succinic Acid Diethyl Ester SCHEMBL22780 0.63 GAA (0.67) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
Succinic Acid Diethyl Ester SCHEMBL27768067 0.63 GAA (0.67) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
SCHEMBL14409745 0.62 TSHR (0.50) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
SCHEMBL1027353 0.62 PPARG (0.36) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
Succinic Acid Diethyl Ester SCHEMBL29494609 0.61 GAA (0.63) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
Succinic Acid Diethyl Ester SCHEMBL21815758 0.61 GAA (0.63) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT
Succinic Acid Diethyl Ester SCHEMBL4324913 0.61 GAA (0.63) SMN1; SMN2CYP4F2CYP4A11ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed