SCHEMBL6565807

SCHEMBL6565807

CC(C)CC(OC(=O)NCc1ccccc1)C(=O)NCC(C#N)COCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.48
CTSL P07711 8/20 0.48
CTSK P43235 6/20 0.48
CTSB P07858 1/20 0.44
PSMB1 P20618 2/20 0.41
PSMB11 A5LHX3 1/20 0.41
PSMD11 O00231 1/20 0.41
PSMD12 O00232 1/20 0.41
PSMD14 O00487 1/20 0.41
PSMA7 O14818 1/20 0.41
PSMD3 O43242 1/20 0.41
PSMC3 P17980 1/20 0.41
PSMA1 P25786 1/20 0.41
PSMA2 P25787 1/20 0.41
PSMA3 P25788 1/20 0.41
PSMA4 P25789 1/20 0.41
PSMB8 P28062 1/20 0.41
PSMB9 P28065 1/20 0.41
PSMA5 P28066 1/20 0.41
PSMB4 P28070 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3907310 0.85 CTSS (0.64) CTSSCTSLCTSKCTSB
SCHEMBL7438088 0.85 CTSS (0.43) CTSSCTSLCTSKCTSB
SCHEMBL3894949 0.82 CTSS (0.56) CTSSCTSLCTSKCTSB
SCHEMBL3907700 0.80 CTSS (0.46) CTSSCTSLCTSKCTSBPSMB1
SCHEMBL3899392 0.79 CTSL (0.50) CTSSCTSLCTSKCTSB
SCHEMBL3895827 0.78 CTSS (0.43) CTSSCTSLCTSKCTSBPSMB1
SCHEMBL3907693 0.77 CTSS (0.44) CTSSCTSLCTSKCTSBPSMB1
SCHEMBL3895384 0.76 CTSC (0.55) CTSSCTSLCTSKCTSB
SCHEMBL3907304 0.75 CTSS (0.44) CTSSCTSLCTSKCTSBPSMB1
SCHEMBL7310650 0.74 ALDH1A1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed