SCHEMBL6566396

SCHEMBL6566396

COc1ccc(OC2CCCC2)cc1C=O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.50
TUBB1 Q9H4B7 1/20 0.48
PDE4B Q07343 9/20 0.47
PDE4A P27815 8/20 0.47
PDE4C Q08493 7/20 0.47
PDE4D Q08499 7/20 0.47
ALDH1A1 P00352 2/20 0.46
NFE2L2 Q16236 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
POLB P06746 2/20 0.43
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30826663 0.87 TUBB1 (0.45) TUBB1PDE4BALDH1A1KDM4ETSHR
SCHEMBL7418526 0.79 ALDH1A1 (0.63) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL172939 0.78 ALDH1A1 (0.71) TUBB1PDE4BPDE4APDE4CPDE4D
SCHEMBL29392394 0.78 ALDH1A1 (0.71) TUBB1PDE4BPDE4APDE4CPDE4D
SCHEMBL6567753 0.78 PTGS1 (0.48) ALDH1A1TSHRPOLB
SCHEMBL7387277 0.78 KMT2A (0.47) HIF1ATUBB1PDE4BPDE4APDE4C
SCHEMBL2004982 0.76 HRH3 (0.54) ALDH1A1
SCHEMBL30826796 0.75 ALDH1A1 (0.58) ALDH1A1POLB
SCHEMBL1665185 0.75 ALDH1A1 (0.47) ALDH1A1NFE2L2KDM4ETDP1
SCHEMBL24750325 0.75 ALDH1A1 (0.56) HIF1APDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135360-B1 NOVEL 3-ALKOXYBENZYLAMINE DERIVATIVES AND THEIR USE AS MEDICINES FOR TREATING SCHIZOPHRENIA PF MEDICAMENT (FR) 2004-03-31 EP disclosed
US-6350913-B1 AROMATIC AMINE COMPOUNDS PIERRE FABRE MEDICAMENT (FR) 2002-02-26 US disclosed
EP-1135360-A1 NOVEL 3-ALKOXYBENZYLAMINE DERIVATIVES AND THEIR USE AS MEDICINES FOR TREATING SCHIZOPHRENIA PIERRE FABRE MEDICAMENT (FR) 2001-09-26 EP disclosed
WO-2000032557-A1 NOVEL 3-ALKOXYBENZYLAMINE DERIVATIVES AND THEIR USE AS MEDICINES FOR TREATING SCHIZOPHRENIA PIERRE FABRE MEDICAMENT (FR) 2000-06-08 WO disclosed