SCHEMBL6566798

SCHEMBL6566798

NC(=O)c1cccc(OCCCN(CC(c2ccccc2)C2CCCCC2)C2CCN(C(=O)O)C(Cc3ccccc3)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 3/20 0.45
PARP14 Q460N5 1/20 0.37
OPRK1 P41145 7/20 0.37
OPRM1 P35372 5/20 0.36
OPRD1 P41143 4/20 0.36
TACR1 P25103 1/20 0.36
KCNH2 Q12809 6/20 0.36
AGTR2 P50052 1/20 0.35
MET P08581 1/20 0.35
FKBP1A P62942 3/20 0.35
CCR5 P51681 1/20 0.35
FKBP5 Q13451 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6513607 0.91 NR1H3 (0.46) NR1H3TACR1AGTR2FKBP1ACCR5
SCHEMBL6564837 0.90 NR1H3 (0.53) NR1H3OPRK1OPRM1OPRD1TACR1
SCHEMBL6567185 0.88 NR1H3 (0.43) NR1H3OPRK1OPRM1OPRD1KCNH2
SCHEMBL6515545 0.86 NR1H3 (0.44) NR1H3PARP14OPRK1OPRM1OPRD1
SCHEMBL6515253 0.86 OPRK1 (0.51) NR1H3OPRK1OPRM1OPRD1KCNH2
SCHEMBL6515170 0.84 NR1H3 (0.44) NR1H3PARP14OPRK1OPRM1OPRD1
SCHEMBL6512055 0.83 NR1H3 (0.45) NR1H3PARP14OPRK1OPRM1OPRD1
SCHEMBL6519566 0.83 NR1H3 (0.42) NR1H3OPRK1OPRM1OPRD1MET
SCHEMBL6567271 0.82 NR1H3 (0.52) NR1H3OPRK1OPRM1OPRD1KCNH2
SCHEMBL6519456 0.81 NR1H3 (0.43) NR1H3OPRM1KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318976-B1 SUBSTITUTED AMINOPROPOXYARYL DERIVATIVES USEFUL AS AGONISTS FOR LXR GLAXO GROUP LTD (GB) 2004-11-24 EP claimed