SCHEMBL6567185

SCHEMBL6567185

CC(C)(C)C1CC(N(CCCOc2cccc(C(N)=O)c2)CC(c2ccccc2)C2CCCCC2)CCN1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 3/20 0.43
OPRK1 P41145 9/20 0.36
KCNH2 Q12809 7/20 0.36
OPRM1 P35372 5/20 0.36
OPRD1 P41143 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
RXRA P19793 1/20 0.34
NR1H2 P55055 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
ESR1 P03372 1/20 0.34
SLC6A4 P31645 1/20 0.34
FFAR1 O14842 1/20 0.34
AGTR2 P50052 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566798 0.88 NR1H3 (0.45) NR1H3OPRK1KCNH2OPRM1OPRD1
SCHEMBL6515545 0.87 NR1H3 (0.44) NR1H3OPRK1KCNH2OPRM1OPRD1
SCHEMBL6512055 0.84 NR1H3 (0.45) NR1H3OPRK1KCNH2OPRM1OPRD1
SCHEMBL6564859 0.84 NR1H3 (0.42) NR1H3MEN1KMT2AHRH3SLC6A4
SCHEMBL6515170 0.83 NR1H3 (0.44) NR1H3OPRK1KCNH2OPRM1OPRD1
SCHEMBL6519456 0.82 NR1H3 (0.43) NR1H3KCNH2OPRM1ALDH1A1HRH3
SCHEMBL6515253 0.82 OPRK1 (0.51) NR1H3OPRK1KCNH2OPRM1OPRD1
SCHEMBL6566799 0.80 NR1H3 (0.54) NR1H3MEN1KMT2AALDH1A1RXRA
SCHEMBL6519566 0.80 NR1H3 (0.42) NR1H3OPRK1OPRM1OPRD1ALDH1A1
SCHEMBL6567271 0.80 NR1H3 (0.52) NR1H3OPRK1KCNH2OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318976-B1 SUBSTITUTED AMINOPROPOXYARYL DERIVATIVES USEFUL AS AGONISTS FOR LXR GLAXO GROUP LTD (GB) 2004-11-24 EP claimed