SCHEMBL6566895

SCHEMBL6566895

Cc1ccc(NC(=O)Nc2c(C)cccc2C)c(O)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.66
KMT2A Q03164 4/20 0.55
MEN1 O00255 1/20 0.55
RAB9A P51151 3/20 0.49
MAPT P10636 2/20 0.49
GBA1 P04062 1/20 0.49
GAA P10253 2/20 0.49
LPAR1 Q92633 1/20 0.48
S1PR4 O95977 1/20 0.48
ALDH1A1 P00352 1/20 0.48
NPC1 O15118 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
LMNA P02545 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TP53 P04637 1/20 0.47
CXCR1 P25024 1/20 0.47
DDX3X O00571 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341663 0.89 CXCR1 (0.59) CXCR2KMT2ARAB9AMAPTALDH1A1
SCHEMBL6567648 0.86 CXCR2 (0.72) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL5195764 0.82 KMT2A (0.64) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL5595504 0.80 CXCR1 (0.66) CXCR2KMT2AMEN1MAPTALDH1A1
SCHEMBL5605320 0.79 CXCR2 (1.00) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL30051979 0.79 MAPT (0.67) KMT2AMEN1RAB9AMAPTGAA
SCHEMBL11575411 0.78 RAB9A (0.60) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL6568502 0.78 RAB9A (0.68) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL5595289 0.77 CXCR1 (0.73) CXCR2KMT2AMEN1RAB9AMAPT
SCHEMBL6436269 0.77 MEN1 (0.72) CXCR2KMT2AMEN1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed