SCHEMBL6567648

SCHEMBL6567648

Cc1ccc(NC(=O)Nc2ccccc2C)c(O)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.72
KMT2A Q03164 2/20 0.60
MEN1 O00255 1/20 0.60
DDX3X O00571 2/20 0.59
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
POLB P06746 3/20 0.55
HTT P42858 2/20 0.55
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.53
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
HSD17B10 Q99714 2/20 0.51
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
TP53 P04637 2/20 0.51
GAA P10253 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347676 0.87 CXCR1 (0.68) CXCR2KMT2AMEN1DDX3XCA12
SCHEMBL6566895 0.86 CXCR2 (0.66) CXCR2KMT2AMEN1DDX3XPOLB
SCHEMBL5595289 0.84 CXCR1 (0.73) CXCR2KMT2AMEN1POLBHTT
SCHEMBL5605320 0.84 CXCR2 (1.00) CXCR2KMT2AMEN1DDX3XHTT
SCHEMBL1275926 0.82 RAB9A (0.75) KMT2AMEN1DDX3XPOLBHTT
SCHEMBL6568502 0.82 RAB9A (0.68) CXCR2KMT2AMEN1CA12CA1
SCHEMBL27576146 0.82 CXCR2 (0.69) CXCR2KMT2AMEN1CA12CA1
SCHEMBL3710548 0.81 CXCR2 (0.71) CXCR2DDX3XCA12CA1CA2
SCHEMBL5852144 0.80 LPAR1 (0.71) KMT2AMEN1DDX3XPOLBALDH1A1
SCHEMBL5594962 0.80 MEN1 (0.72) CXCR2KMT2AMEN1DDX3XCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed