SCHEMBL6567204

SCHEMBL6567204

COc1cc(CNC(=O)c2ccccc2C(F)(F)F)ccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.53
PTPN7 P35236 1/20 0.52
DUSP3 P51452 1/20 0.52
HPGD P15428 4/20 0.51
TP53 P04637 1/20 0.51
GLA P06280 1/20 0.51
APEX1 P27695 1/20 0.51
GABRP O00591 1/20 0.51
GABRD O14764 1/20 0.51
GABRA1 P14867 1/20 0.51
GABRB1 P18505 1/20 0.51
GABRG2 P18507 1/20 0.51
GABRB3 P28472 1/20 0.51
GABRA5 P31644 1/20 0.51
GABRA3 P34903 1/20 0.51
GABRA2 P47869 1/20 0.51
GABRB2 P47870 1/20 0.51
GABRA4 P48169 1/20 0.51
GABRE P78334 1/20 0.51
GABRA6 Q16445 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031773 0.85 TRPV1 (0.59) TRPV1HPGDTP53GLAAPEX1
SCHEMBL14698338 0.82 APEX1 (0.59) TRPV1HPGDTP53GLAAPEX1
SCHEMBL30520585 0.81 APEX1 (0.58) TRPV1HPGDTP53GLAAPEX1
SCHEMBL21623922 0.81 APEX1 (0.58) TRPV1HPGDTP53GLAAPEX1
SCHEMBL5681720 0.79 ERCC1 (0.69) TRPV1PTPN7DUSP3SMN1; SMN2
SCHEMBL30386504 0.78 APEX1 (0.56) TRPV1HPGDTP53GLAAPEX1
SCHEMBL3455177 0.77 LMNA (0.54) HPGDAPEX1LMNAALDH1A1CYP1A2
SCHEMBL7715505 0.77 DUSP3 (0.65) PTPN7DUSP3SMN1; SMN2
SCHEMBL898313 0.77 PTPN7 (0.54) PTPN7DUSP3HPGDALDH1A1CYP1A2
SCHEMBL5065598 0.76 NR1H4 (0.64) PTPN7DUSP3HPGDLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed