SCHEMBL6567375

SCHEMBL6567375

O=S(=O)(NCc1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.74
LMNA P02545 2/20 0.70
RAB9A P51151 1/20 0.70
KEAP1 Q14145 1/20 0.63
NAMPT P43490 1/20 0.57
TRPV1 Q8NER1 1/20 0.56
PPARG P37231 1/20 0.53
KAT6A Q92794 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
MMP1 P03956 1/20 0.51
MMP2 P08253 1/20 0.51
MMP9 P14780 1/20 0.51
MMP8 P22894 1/20 0.51
MMP13 P45452 1/20 0.51
CA12 O43570 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
ATM Q13315 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30927212 1.00 CYP19A1 (0.74) CYP19A1LMNARAB9AKEAP1NAMPT
SCHEMBL20946446 0.87 CYP19A1 (0.72) CYP19A1LMNARAB9ANAMPTTRPV1
SCHEMBL13888909 0.85 KEAP1 (0.63) CYP19A1LMNARAB9AKEAP1SMN1; SMN2
SCHEMBL21048461 0.84 KEAP1 (0.81) CYP19A1LMNAKEAP1SMN1; SMN2CA1
SCHEMBL14094673 0.84 CYP19A1 (0.67) CYP19A1LMNARAB9ANAMPTTRPV1
SCHEMBL14129032 0.84 CYP19A1 (0.67) CYP19A1LMNARAB9ANAMPTTRPV1
SCHEMBL22489364 0.83 CYP19A1 (0.63) CYP19A1LMNARAB9ANAMPTTRPV1
SCHEMBL1954496 0.83 CYP19A1 (0.80) CYP19A1LMNARAB9AKEAP1NAMPT
SCHEMBL3853891 0.83 CYP19A1 (0.70) CYP19A1LMNARAB9AKEAP1NAMPT
SCHEMBL13972872 0.83 CYP19A1 (0.66) CYP19A1LMNARAB9ANAMPTTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103588697-B Disubstituted benzenes sulfamide compound of one class 2,5 and its production and use 中国科学院上海药物研究所 2017-09-15 CN claimed
CN-103588697-B Disubstituted benzenes sulfamide compound of one class 2,5 and its production and use 中国科学院上海药物研究所 2017-09-15 CN disclosed
CN-102802731-A Benzimidazole derivatives useful as TRPM8 channel modulators JANSSEN PHARMACEUTICA NV 2012-11-28 CN disclosed
EP-1443041-A1 5-AMIDINO-2-HYDROXYBENZENESULFONAMIDE DERIVATIVES, MEDICINAL COMPOSITIONS CONTAINING THE SAME, MEDICINAL USE THEREOF AND INTERMEDIATES IN THE PRODUCTION THEREOF Kissei Pharmaceutical Co., Ltd. (JP) 2004-08-04 EP disclosed