SCHEMBL6567652

SCHEMBL6567652

O=C(Nc1cc(Cl)c(O)c(Cl)c1)Nc1ccc2ccccc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.66
RAB9A P51151 6/20 0.66
MAPT P10636 6/20 0.66
GRIK1 P39086 1/20 0.56
GRIK2 Q13002 1/20 0.56
CA2 P00918 2/20 0.55
CNR1 P21554 1/20 0.55
EPHX1 P07099 1/20 0.54
EPHX2 P34913 1/20 0.54
MEN1 O00255 7/20 0.54
KMT2A Q03164 7/20 0.54
TDP1 Q9NUW8 1/20 0.54
GAA P10253 2/20 0.54
KDM4E B2RXH2 1/20 0.54
KDR P35968 1/20 0.53
POLB P06746 2/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA9 Q16790 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547503 0.85 RAB9A (0.89) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL11057371 0.82 NPC1 (0.77) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL4342381 0.82 KMT2A (0.68) NPC1RAB9AMAPTCNR1EPHX1
SCHEMBL6567241 0.81 EPHX1 (0.59) NPC1RAB9AMAPTCA2EPHX1
SCHEMBL24272500 0.80 MAPT (0.80) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL24272501 0.80 MAPT (0.80) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL12846485 0.80 DEGS1 (0.66) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL11049543 0.80 MAPT (1.00) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL30697002 0.80 MAPT (1.00) NPC1RAB9AMAPTGRIK1GRIK2
SCHEMBL3668804 0.79 CNR1 (0.61) NPC1RAB9AMAPTGRIK1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed