SCHEMBL6568415

SCHEMBL6568415

CC(=O)NOP(=O)(O)OCCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
CA9 Q16790 1/20 0.42
ALDH1A1 P00352 2/20 0.41
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ANPEP P15144 2/20 0.40
ERAP1 Q9NZ08 2/20 0.40
ERAP2 Q6P179 1/20 0.40
S1PR4 O95977 1/20 0.39
S1PR1 P21453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6570293 0.86 POLB (0.48) TSHRNPC1RAB9ACA12CA1
SCHEMBL6570112 0.86 TSHR (0.41) TSHRNPC1RAB9ACA12CA1
SCHEMBL6568406 0.85 NPC1 (0.50) TSHRNPC1RAB9ACA12CA1
SCHEMBL6568562 0.83 HDAC3 (0.44) TSHRNPC1RAB9AESR1ESR2
SCHEMBL6571631 0.83 GAA (0.43) TSHRLMNAKDM4ECYP3A4HPGD
SCHEMBL6569361 0.83 MTNR1A (0.53) CA1CA2CA9ALDH1A1KDM4E
SCHEMBL6569232 0.82 CA12 (0.43) TSHRCA12CA1ANPEPERAP1
SCHEMBL6570330 0.81 TDP1 (0.46) NPC1RAB9ALMNAKDM4EHPGD
SCHEMBL6569921 0.81 HDAC1 (0.51) TSHRLMNA
SCHEMBL6570338 0.81 ALDH1A1 (0.41) TSHRNPC1RAB9ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1156054-B1 DRUGS CONTAINING PHOSPHORIC ACID DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-04-14 EP claimed
US-6495533-B1 TUMOR NECROSIS FACTOR INHIBITORS; RHEUMATOID ARTHRITIS, ULCERATIVE COLITIS, CROHN'S DISEASE, HEPATITIS, SEPSIS, HEMORRHAGIC SHOCK, MULTIPLE SCLEROSIS, CEREBRAL INFARCTION, DIABETES, INTERSTITIAL PNEUMONIA, PAIN, HIV ONO PHARMACEUTICAL CO., LTD. (JP) 2002-12-17 US claimed
EP-1156054-A1 DRUGS CONTAINING PHOSPHORIC ACID DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-11-21 EP claimed