SCHEMBL6568642

SCHEMBL6568642

CC(C)(C)c1nc(-c2cc(Cl)c(O)c(Cl)c2)cs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.43
COMT P21964 1/20 0.43
TTR P02766 1/20 0.41
CNR1 P21554 5/20 0.39
MAPT P10636 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
RECQL P46063 1/20 0.37
ESR2 Q92731 1/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
ABL1 P00519 4/20 0.37
ALOX5 P09917 1/20 0.36
VCP P55072 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19625347 0.87 COMT (0.39) CNR2COMTCNR1MAPTGAA
SCHEMBL6565664 0.81 GAA (0.56) TTRMAPTGAAKDM4EALDH1A1
SCHEMBL13650700 0.81 CYP1A2 (0.53) MAPTKDM4EABL1ALOX5VCP
SCHEMBL6568655 0.78 CNR2 (0.50) CNR2TTRCNR1MAPTGAA
SCHEMBL19625313 0.77 ABL1 (0.55) CNR2COMTCNR1MAPTALDH1A1
SCHEMBL19625311 0.75 MAPT (0.50) MAPTGAAKDM4EALDH1A1RECQL
SCHEMBL19625348 0.75 COMT (0.34) COMTMAPTALDH1A1ALOX5MEN1
SCHEMBL12282347 0.75 LTA4H (0.58) COMTMAPTGAAKDM4EALDH1A1
SCHEMBL799889 0.75 RAB9A (0.56) MAPTGAAKDM4EALDH1A1POLB
SCHEMBL19625338 0.74 ABL1 (0.55) CNR2COMTMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed