SCHEMBL6568332

SCHEMBL6568332

CN(C)C(=O)Oc1ccc(C[C@H](NC(=O)[C@@H]2OC(=O)N[C@H]2Cc2ccccc2)C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 20/20 0.47
ITGB1 P05556 19/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6568255 0.87 LMNA (0.46) ITGA4
SCHEMBL6568258 0.87 LMNA (0.46) ITGA4
SCHEMBL7224758 0.87 LMNA (0.46) ITGA4
SCHEMBL6568912 0.75 ITGB1 (0.51) ITGA4ITGB1
SCHEMBL7222897 0.73 ACACB (0.43)
SCHEMBL7401957 0.72 ITGB1 (0.43) ITGA4ITGB1
SCHEMBL5679669 0.72 ITGB1 (0.63) ITGA4ITGB1
SCHEMBL5681731 0.71 ITGA4 (0.43) ITGA4ITGB1
SCHEMBL13841280 0.70 ITGB1 (0.57) ITGA4ITGB1
SCHEMBL12834784 0.69 ITGA4 (0.44) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161416-B1 ALPHA-AMINOACETIC ACID DERIVATIVES USEFUL AS ALPHA 4 BETA 7 - RECEPTOR ANTAGONISTS ELAN PHARM INC (US) 2004-04-14 EP claimed
US-6545160-B2 Alpha-aminoacetic acid derivatives bind alpha 4 beta 7 integrin, useful for treatment of inflammatory diseases in mammalian patient, such as asthma, Alzheimer's disease, atherosclerosis, AIDS dementia, diabetes, rheumatoid arthritis ELAN PHARMACEUTICALS, INC. 2003-04-08 US disclosed