SCHEMBL6569728

SCHEMBL6569728

COC(=O)c1ccc(NC(=O)C(C)(O)C(F)(F)F)c(OC)c1

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 5/20 0.74
ABCC8 Q09428 5/20 0.74
KCNJ11 Q14654 5/20 0.74
KCNJ8 Q15842 5/20 0.74
PDK1 Q15118 12/20 0.73
PDK2 Q15119 12/20 0.73
PDK3 Q15120 12/20 0.73
PDK4 Q16654 12/20 0.73
NR1H2 P55055 1/20 0.53
NR1H3 Q13133 1/20 0.53
TSHR P16473 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
PYGL P06737 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607928 0.85 ABCC9 (1.00) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6347722 0.84 PDK1 (0.73) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6569428 0.84 TSHR (0.71) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6351244 0.83 PDK1 (0.71) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6569716 0.83 PDK1 (0.67) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6569709 0.83 PDK1 (0.67) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6567832 0.80 PDK1 (0.66) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6567827 0.80 PDK1 (0.66) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL6350417 0.79 PDK1 (1.00) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL15693330 0.77 ALDH1A1 (0.62) PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed