SCHEMBL6570808

SCHEMBL6570808

COC(=O)CCNC(=O)c1cc(N2CC2)c([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.54
CYP3A4 P08684 2/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
NPC1 O15118 1/20 0.46
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
ALDH1A1 P00352 5/20 0.44
SIRT6 Q8N6T7 2/20 0.43
POLB P06746 1/20 0.43
RECQL P46063 1/20 0.42
HDAC1 Q13547 1/20 0.41
LMNA P02545 4/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6573690 0.81 CYP3A4 (0.50) MAPTCYP3A4NPC1ALDH1A1POLB
SCHEMBL6569993 0.77 LMNA (0.68) MAPTCYP3A4BLMPMP22DRD2
SCHEMBL6572262 0.76 SMN1; SMN2 (0.69) MAPTCYP3A4BLMPMP22ALDH1A1
SCHEMBL366651 0.75 MAPT (0.55) MAPTCYP3A4BLMPMP22NPC1
SCHEMBL6573702 0.75 MAPT (0.59) MAPTCYP3A4BLMPMP22NPC1
SCHEMBL6573527 0.75 SMN1; SMN2 (0.65) MAPTCYP3A4BLMPMP22ALDH1A1
SCHEMBL8761909 0.74 NPC1 (0.44) MAPTCYP3A4NPC1ALDH1A1POLB
SCHEMBL11120951 0.72 MAPT (0.74) MAPTCYP3A4BLMPMP22ALDH1A1
SCHEMBL2977898 0.71 MEN1 (0.44) MAPTCYP3A4NPC1ALDH1A1POLB
Hydrochloric Acid SCHEMBL9251441 0.71 LMNA (0.43) MAPTCYP3A4NPC1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6517836-B1 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes AUCKLAND UNISERVICES LIMITED (NZ) 2003-02-11 US claimed
EP-1109550-B1 NOVEL NITROPHENYLAZIRIDINE COMPOUNDS AND THEIR USE AS PRODRUGS AUCKLAND UNISERVICES LTD (NZ) 2004-11-24 EP disclosed
US-6517836-B1 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes AUCKLAND UNISERVICES LIMITED (NZ) 2003-02-11 US disclosed