SCHEMBL6573527

SCHEMBL6573527

O=C(NCCCCN1CCOCC1)c1cc(N2CC2)c([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.65
LMNA P02545 8/20 0.64
ALDH1A1 P00352 2/20 0.63
GAA P10253 1/20 0.63
CYP2C19 P33261 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
MAOB P27338 1/20 0.51
MAPT P10636 3/20 0.49
CYP3A4 P08684 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
RAB9A P51151 1/20 0.49
TSHR P16473 1/20 0.47
HDAC1 Q13547 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572262 0.97 SMN1; SMN2 (0.69) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL6569993 0.93 LMNA (0.68) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL6571185 0.86 LMNA (0.71) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL6570770 0.83 LMNA (0.76) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL6573530 0.78 CYP2C19 (0.74) SMN1; SMN2LMNAALDH1A1CYP2C19L3MBTL1
SCHEMBL28677732 0.78 SMN1; SMN2 (0.63) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL9246238 0.78 LMNA (0.72) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL6573581 0.76 MAPT (0.50) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL27672667 0.76 LMNA (0.66) SMN1; SMN2LMNAALDH1A1GAACYP2C19
SCHEMBL2969374 0.75 SMN1; SMN2 (0.74) SMN1; SMN2LMNAALDH1A1GAACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6517836-B1 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes AUCKLAND UNISERVICES LIMITED (NZ) 2003-02-11 US claimed
EP-1109550-B1 NOVEL NITROPHENYLAZIRIDINE COMPOUNDS AND THEIR USE AS PRODRUGS AUCKLAND UNISERVICES LTD (NZ) 2004-11-24 EP disclosed
US-6517836-B1 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes AUCKLAND UNISERVICES LIMITED (NZ) 2003-02-11 US disclosed