SCHEMBL6571083

SCHEMBL6571083

CNc1ccc(N)c(-c2ccc(N)cc2N)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.38
HTR6 P50406 3/20 0.34
PDK2 Q15119 1/20 0.31
GLA P06280 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.30
RPS6KA2 Q15349 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6570907 0.90 HTR6 (0.37) CASP1HTR6POLBTSHRALDH1A1
SCHEMBL6571922 0.86 TSHR (0.41) CASP1HTR6PDK2POLBGAA
SCHEMBL6572813 0.82 PRKCI (0.34) CASP1HTR6GLAPOLBGAA
SCHEMBL6572508 0.82 HTR6 (0.33) CASP1HTR6POLBTSHRALDH1A1
SCHEMBL3790053 0.81 ALDH1A1 (0.52) CASP1PDK2GLAGAATSHR
SCHEMBL6570909 0.81 PDE10A (0.44) CASP1HTR6POLBGAATSHR
SCHEMBL5900560 0.80 KDM4E (0.41) CASP1GAAALDH1A1
SCHEMBL6011526 0.80 CASP1 (0.44) CASP1GLAPOLBGAATSHR
SCHEMBL3790061 0.79 HTR6 (0.39) HTR6TSHRALDH1A1
SCHEMBL3784065 0.77 ALDH1A1 (0.52) CASP1PDK2GLAGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed