SCHEMBL6571104

SCHEMBL6571104

COCCNc1ccc(N)cc1-c1c(OC)cccc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.42
NCF1 P14598 2/20 0.41
ALDH1A1 P00352 6/20 0.39
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 3/20 0.39
LMNA P02545 3/20 0.39
CYP2C19 P33261 2/20 0.39
HSD17B10 Q99714 3/20 0.38
MAPK1 P28482 3/20 0.38
KDM4E B2RXH2 2/20 0.38
CYP2D6 P10635 2/20 0.38
USP2 O75604 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPT P10636 4/20 0.37
TSHR P16473 2/20 0.37
CLK4 Q9HAZ1 1/20 0.37
NR3C1 P04150 1/20 0.37
GAA P10253 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572270 0.86 ALDH1A1 (0.50) PTGER4NCF1ALDH1A1CYP1A2CYP3A4
SCHEMBL6571037 0.86 TSHR (0.40) ALDH1A1MAPK1KDM4EUSP2MAPT
SCHEMBL6570689 0.82 PTGER4 (0.48) PTGER4NCF1ALDH1A1LMNAKDM4E
SCHEMBL6572456 0.81 PTGER4 (0.50) PTGER4NCF1ALDH1A1CYP1A2LMNA
SCHEMBL9499986 0.81 PTGER4 (0.49) PTGER4NCF1ALDH1A1LMNAMAPK1
SCHEMBL6570803 0.80 PTGER4 (0.41) PTGER4NCF1ALDH1A1LMNAHSD17B10
SCHEMBL6572605 0.80 APP (0.43) ALDH1A1CYP3A4LMNAMAPK1KDM4E
SCHEMBL6571332 0.80 CYP1A2 (0.49) PTGER4NCF1ALDH1A1CYP1A2CYP3A4
SCHEMBL6571509 0.79 CYP3A4 (0.46) PTGER4NCF1ALDH1A1CYP1A2CYP3A4
SCHEMBL6572446 0.79 PTGER4 (0.40) PTGER4NCF1ALDH1A1MAPTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed