SCHEMBL6572405

SCHEMBL6572405

COc1ccc(OC)c(-c2cc(N)ccc2N(CCO)CCO)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
GABRG2 P18507 5/20 0.39
GABRB3 P28472 5/20 0.39
GABRA2 P47869 5/20 0.39
ALDH1A1 P00352 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
THRB P10828 1/20 0.39
ADRA1A P35348 3/20 0.38
TAAR1 Q96RJ0 1/20 0.38
AOC3 Q16853 1/20 0.38
CYP19A1 P11511 1/20 0.37
DHFR P00374 1/20 0.37
ADRA2A P08913 2/20 0.37
HTR2A P28223 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107403 0.91 HDAC4 (0.39) HDAC4HDAC2HDAC8GABRG2GABRB3
SCHEMBL6570817 0.87 HDAC4 (0.39) HDAC4HDAC2HDAC8GABRG2GABRB3
SCHEMBL6570737 0.86 MEN1 (0.47) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL6571296 0.86 GAA (0.40) ALDH1A1MEN1KMT2AMAPTTHRB
SCHEMBL6571978 0.84 HTR7 (0.41) MEN1KMT2AMAPTHTR2A
SCHEMBL6571974 0.84 ALDH1A1 (0.42) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL6571940 0.83 ALDH1A1 (0.42) ALDH1A1CYP19A1KDM4EHPGD
SCHEMBL6570844 0.83 TRIM24 (0.42) HDAC8ALDH1A1CYP19A1KDM4ENPC1
SCHEMBL6573059 0.82 HDAC4 (0.40) HDAC4HDAC2HDAC8ALDH1A1MAPT
SCHEMBL6570775 0.81 ERN1 (0.42) ALDH1A1MEN1KMT2AMAPTCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed