SCHEMBL6573092

SCHEMBL6573092

O=[N+]([O-])c1ccc(F)c(-c2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.55
ALDH1A1 P00352 4/20 0.55
HIF1A Q16665 1/20 0.55
RAB9A P51151 3/20 0.54
POLB P06746 1/20 0.54
PTGDR2 Q9Y5Y4 1/20 0.52
PTPRC P08575 3/20 0.50
S100A4 P26447 2/20 0.50
NPC1 O15118 2/20 0.50
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
CES1 P23141 1/20 0.50
LMNA P02545 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MAPT P10636 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
MYC P01106 1/20 0.47
MAX P61244 1/20 0.47
CYP19A1 P11511 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10684532 0.86 RAB9A (0.58) PTGS2ALDH1A1HIF1ARAB9APOLB
SCHEMBL4910527 0.85 ALDH1A1 (0.67) ALDH1A1HIF1APTPRCS100A4BCHE
SCHEMBL6391559 0.83 PTGS2 (0.69) PTGS2ALDH1A1RAB9APOLBPTGDR2
SCHEMBL28207049 0.83 PTGS2 (0.73) PTGS2ALDH1A1RAB9APOLBPTGDR2
SCHEMBL1931406 0.83 ALDH1A1 (0.51) PTGS2ALDH1A1HIF1APTPRCS100A4
SCHEMBL9568408 0.83 ALDH1A1 (0.55) PTGS2ALDH1A1HIF1ARAB9APOLB
SCHEMBL2650165 0.83 MAPK14 (0.52) ALDH1A1HIF1ARAB9APOLBPTPRC
SCHEMBL9568330 0.82 TDP1 (0.59) ALDH1A1HIF1APOLBPTGDR2CES1
SCHEMBL10516385 0.82 ALDH1A1 (0.47) PTGS2ALDH1A1HIF1ARAB9APOLB
SCHEMBL10518694 0.82 TP53 (0.60) ALDH1A1RAB9APOLBNPC1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103958500-B Kinases inhibitor ORION CORP. (FI) 2016-04-27 CN disclosed
CN-105283443-A Heterocyclic derivatives and use thereof C & C RES LAB 2016-01-27 CN disclosed
CN-1303043-C Process for producing biaryl compound SUMITOMO CHEMICAL CO (JP) 2007-03-07 CN disclosed
CN-1642879-A Process for preparing diaryl compounds SUMITOMO CHEMICAL CO (JP) 2005-07-20 CN disclosed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed
EP-0184384-B1 SUBSTITUTED DIHYDROQUINOLONE CARBOXYLIC ACIDS, ANTI-BACTERIAL COMPOSITIONS CONTAINING THEM PFIZER INC. (US) 1989-08-02 EP disclosed
US-4623650-A BACTERICIDES PFIZER INC. (US) 1986-11-18 US disclosed
EP-0184384-A1 Substituted dihydroquinolone carboxylic acids, anti-bacterial compositions containing them PFIZER INC. (US) 1986-06-11 EP disclosed