SCHEMBL6573875

SCHEMBL6573875

COc1ccc(OC)c(-c2cc(N)ccc2NCC(O)CO)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.39
ADRA2A P08913 2/20 0.39
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
TSHR P16473 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
KMT2A Q03164 2/20 0.36
AR P10275 1/20 0.36
VDR P11473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
KCNA5 P22460 1/20 0.36
KCNH2 Q12809 1/20 0.36
ALDH1A1 P00352 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7686147 0.91 RPS6KA2 (0.40) ADRA1AADRA2AADRB2ADRB1ADRB3
SCHEMBL6570673 0.86 AGTR1 (0.42) LMNACYP1A2KMT2AALDH1A1MAPK1
SCHEMBL6570661 0.85 RPS6KA2 (0.40) TSHRCYP1A2CYP2C19KMT2AKCNA5
SCHEMBL6572048 0.84 AR (0.36) ARVDRHDAC4HDAC2HDAC8
SCHEMBL6572745 0.83 RAD52 (0.41) ADRA1AKMT2AHDAC4HDAC2HDAC8
SCHEMBL6571130 0.82 TSHR (0.38) TSHRARVDRKCNA5KCNH2
SCHEMBL6572994 0.81 TSHR (0.44) TSHRLMNAKCNA5KCNH2ALDH1A1
SCHEMBL6573393 0.81 AGTR1 (0.39) TSHRLMNACYP1A2KMT2AAR
SCHEMBL6572446 0.78 PTGER4 (0.40) ADRA1AKMT2ANPSR1HDAC4HDAC2
SCHEMBL6571210 0.77 ALDH1A1 (0.45) ADRA1ATSHRLMNAKMT2AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed