SCHEMBL6571130

SCHEMBL6571130

COc1cc(OC)cc(-c2cc(N)ccc2NCC(O)CO)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
ABL1 P00519 2/20 0.37
ABCB1 P08183 2/20 0.37
BCR P11274 2/20 0.37
KIT P10721 1/20 0.36
KCNA5 P22460 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP19A1 P11511 2/20 0.35
RPS6KA2 Q15349 1/20 0.34
AR P10275 2/20 0.34
VDR P11473 2/20 0.34
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
NQO2 P16083 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6570661 0.91 RPS6KA2 (0.40) TSHRMAPK1KITKCNA5KCNH2
SCHEMBL6572994 0.89 TSHR (0.44) TSHRMAPK1KITKCNA5KCNH2
SCHEMBL6572042 0.85 PDE3B (0.34) ARVDR
SCHEMBL6574847 0.84 PDE3B (0.37) ARVDR
SCHEMBL7686147 0.82 RPS6KA2 (0.40) TSHRMAPK1KCNA5KCNH2RPS6KA2
SCHEMBL6573875 0.82 ADRA1A (0.39) TSHRMAPK1KCNA5KCNH2AR
SCHEMBL6571431 0.82 AR (0.36) TSHRARVDRGAAMAPT
SCHEMBL6572447 0.82 ADRB2 (0.33) ABL1ABCB1BCRARVDR
SCHEMBL6572442 0.82 ABL1 (0.40) TSHRMAPK1ABL1ABCB1BCR
SCHEMBL6573393 0.81 AGTR1 (0.39) TSHRMAPK1ARVDRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed