SCHEMBL6574304

SCHEMBL6574304

COc1ccc(CSC(C)(C)C(=O)NCCN(CCNCCN)C(=O)C(C)(C)SCc2ccc(OC)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.36
GAA P10253 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
DRD4 P21917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575126 0.87 PPIB (0.40) IDO1GAAPOLBSMN1; SMN2ALDH1A1
SCHEMBL6575543 0.85 MIF (0.35) GAASMN1; SMN2ALDH1A1
SCHEMBL6574310 0.83 CYP1A2 (0.41) IDO1GAAPOLBSMN1; SMN2ALDH1A1
SCHEMBL6575122 0.76 IDO1 (0.40) IDO1GAASMN1; SMN2ALDH1A1
SCHEMBL6575981 0.72 MEN1 (0.54) IDO1GAAPOLBSMN1; SMN2ALDH1A1
SCHEMBL6575055 0.71 OPRK1 (0.37) GAASMN1; SMN2ALDH1A1
SCHEMBL30657036 0.69 TAAR1 (0.44) IDO1GAAPOLBSMN1; SMN2
SCHEMBL27360388 0.69 HTT (0.47) IDO1GAASMN1; SMN2ALDH1A1
SCHEMBL8837514 0.68 MAPT (0.53) GAAPOLBSMN1; SMN2ALDH1A1
SCHEMBL8837485 0.67 MAPT (0.44) GAASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785928-B1 NOVEL N3 S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC (CA) 2004-04-28 EP disclosed
EP-0785951-B1 TC OR RE RADIOLABELLED SOMATOSTATIN ANALOGS MERCK FROSST CANADA INC (CA) 2002-04-24 EP disclosed
US-5632969-A N3 S2 chelating ligands optionally radiolabelled with Tc or Re, useful for diagnostic or therapeutic applications MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5556939-A TC or RE radionuclide labelled chelate, hexapeptide complexes useful for diagnostic or therapeutic applications MERCK FROSST CANADA, INC. (CA) 1996-09-17 US disclosed