SCHEMBL6575543

SCHEMBL6575543

COc1ccc(CSC(C)(C)C(=O)NCCN(CCNCCN=C=S)C(=O)C(C)(C)SCc2ccc(OC)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MIF P14174 1/20 0.35
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP3A4 P08684 1/20 0.31
NAAA Q02083 2/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
KEAP1 Q14145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575057 0.86 MEN1 (0.35) GAASMN1; SMN2ALDH1A1HDAC3HDAC1
SCHEMBL6575545 0.85 CYP1A2 (0.39) MIFGAASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL6574304 0.85 IDO1 (0.36) GAASMN1; SMN2ALDH1A1
SCHEMBL6575126 0.81 PPIB (0.40) GAASMN1; SMN2ALDH1A1HDAC3HDAC1
SCHEMBL6575055 0.76 OPRK1 (0.37) MIFGAASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL6574310 0.72 CYP1A2 (0.41) GAASMN1; SMN2ALDH1A1CYP1A2CYP2D6
SCHEMBL6575523 0.71 ALDH1A1 (0.53) GAASMN1; SMN2ALDH1A1CYP3A4MEN1
SCHEMBL6575122 0.70 IDO1 (0.40) GAASMN1; SMN2ALDH1A1CYP1A2CYP2D6
SCHEMBL6575981 0.68 MEN1 (0.54) GAASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL27360388 0.65 HTT (0.47) GAASMN1; SMN2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785928-B1 NOVEL N3 S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC (CA) 2004-04-28 EP disclosed
EP-0785951-B1 TC OR RE RADIOLABELLED SOMATOSTATIN ANALOGS MERCK FROSST CANADA INC (CA) 2002-04-24 EP disclosed
US-5556939-A TC or RE radionuclide labelled chelate, hexapeptide complexes useful for diagnostic or therapeutic applications MERCK FROSST CANADA, INC. (CA) 1996-09-17 US disclosed