SCHEMBL6575126

SCHEMBL6575126

COc1ccc(CSC(C)(C)C(=O)NCCN(CCNCc2ccc(N)cc2)C(=O)C(C)(C)SCc2ccc(OC)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIB P23284 1/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
IDO1 P14902 2/20 0.36
CHRM2 P08172 1/20 0.36
NPC1 O15118 1/20 0.36
EPHX2 P34913 1/20 0.36
RAB9A P51151 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574304 0.87 IDO1 (0.36) ALDH1A1IDO1POLBSMN1; SMN2GAA
SCHEMBL6575122 0.82 IDO1 (0.40) PPIBALDH1A1IDO1SMN1; SMN2GAA
SCHEMBL6575543 0.81 MIF (0.35) MEN1KMT2AALDH1A1NPC1EPHX2
SCHEMBL6574310 0.77 CYP1A2 (0.41) MEN1KMT2AALDH1A1IDO1NPC1
SCHEMBL6575981 0.70 MEN1 (0.54) MEN1KMT2AALDH1A1IDO1NPC1
SCHEMBL6575055 0.69 OPRK1 (0.37) MEN1KMT2AALDH1A1HDAC3HDAC1
SCHEMBL3900702 0.67 EPHX2 (0.40) PPIBMEN1KMT2AALDH1A1KDM4E
SCHEMBL27360388 0.67 HTT (0.47) MEN1KMT2AALDH1A1IDO1NPC1
SCHEMBL8837514 0.66 MAPT (0.53) MEN1KMT2AALDH1A1KDM4ENPC1
SCHEMBL21066542 0.66 MEN1 (0.54) MEN1KMT2AATMALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785928-B1 NOVEL N3 S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC (CA) 2004-04-28 EP disclosed
EP-0785951-B1 TC OR RE RADIOLABELLED SOMATOSTATIN ANALOGS MERCK FROSST CANADA INC (CA) 2002-04-24 EP disclosed
US-5632969-A N3 S2 chelating ligands optionally radiolabelled with Tc or Re, useful for diagnostic or therapeutic applications MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5556939-A TC or RE radionuclide labelled chelate, hexapeptide complexes useful for diagnostic or therapeutic applications MERCK FROSST CANADA, INC. (CA) 1996-09-17 US disclosed