SCHEMBL6576750

SCHEMBL6576750

CC(C)Nc1ncnc2c1ncn2[C@@H]1O[C@H](c2nc(C(C)(C)C)no2)[C@@H](O)[C@H]1O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DOT1L Q8TEK3 1/20 0.48
ADORA3 P0DMS8 3/20 0.47
ADORA2A P29274 3/20 0.47
ADORA2B P29275 2/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
NFKB1 P19838 1/20 0.47
HIF1A Q16665 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
PMP22 Q01453 1/20 0.47
NPC1 O15118 1/20 0.47
ADORA1 P30542 1/20 0.47
RAB9A P51151 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6576646 0.89 ADORA3 (0.50) ADORA3ADORA2AADORA2BADORA1
SCHEMBL6572956 0.86 ADORA3 (0.58) ADORA3ADORA2AADORA2BTP53TSHR
SCHEMBL6575094 0.85 ADORA3 (0.49) DOT1LADORA3ADORA2AADORA2BTP53
SCHEMBL6574553 0.84 ADORA3 (0.60) ADORA3ADORA2AADORA2BADORA1
SCHEMBL6574608 0.84 ADORA3 (0.59) ADORA3ADORA2AADORA2BTP53TSHR
SCHEMBL6575273 0.82 ADORA3 (0.51) ADORA3ADORA2AADORA2BTP53TSHR
SCHEMBL6576848 0.81 ADORA3 (0.53) ADORA3ADORA2AADORA2BTSHRNFKB1
SCHEMBL6576747 0.81 ADORA3 (0.54) ADORA3ADORA2AADORA2BTSHRNFKB1
SCHEMBL6575274 0.81 ADORA2A (0.51) ADORA3ADORA2AADORA2BTP53TSHR
SCHEMBL6574563 0.81 ADORA3 (0.47) ADORA3ADORA2AADORA2BTSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090019-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2004-09-29 EP disclosed
EP-1447407-A1 Adenosine derivatives GLAXO GROUP LIMITED (GB) 2004-08-18 EP disclosed