SCHEMBL6577070

SCHEMBL6577070

CCCCCCCCOc1c(C=CCO)c2ccc(OCCCC)cc2[nH]c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.48
ALDH2 P05091 1/20 0.39
HTR1A P08908 6/20 0.39
HTR1D P28221 6/20 0.39
HTR1B P28222 6/20 0.39
MAPT P10636 3/20 0.39
MAPK1 P28482 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TP53 P04637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HTR2A P28223 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAOA P21397 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578984 0.89 GPR84 (0.39) GPR17ALDH2MAPTKDM4EMEN1
SCHEMBL6581344 0.89 HTT (0.39) GPR17MAPTKDM4EMEN1KMT2A
SCHEMBL6579789 0.88 PTGES (0.43) GPR17MAPK1TDP1CYP1A2CYP3A4
SCHEMBL6582134 0.82 PARP1 (0.44) MAPTTDP1TP53KDM4EMEN1
SCHEMBL7998930 0.70 PARP1 (0.46) GPR17HTR1AHTR1DHTR1BMAPT
SCHEMBL8004628 0.70 PARP1 (0.46) GPR17HTR1AHTR1DHTR1BMAPT
SCHEMBL8001131 0.70 PARP1 (0.46) GPR17HTR1AHTR1DHTR1BMAPT
SCHEMBL8001153 0.70 AR (0.44) GPR17HTR1AHTR1DHTR1BMAPT
SCHEMBL7988485 0.70 AR (0.44) GPR17HTR1AHTR1DHTR1BMAPT
SCHEMBL7998801 0.70 AR (0.44) GPR17HTR1AHTR1DHTR1BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927718-B1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK & CHEMICALS (JP) 2004-02-25 EP disclosed
US-6271416-B1 O-(HYDROCARBONOXYACETAMIDO)BENZOIC ACID DERIVATIVES AS INTERMEDIATES DAINIPPON INK AND CHEMICALS, INC. (JP) 2001-08-07 US disclosed
US-6136822-A ETHER, HYDROXY QUINOLINONE COMPOUNDS DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-10-24 US disclosed
EP-0927718-A1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-07-07 EP disclosed